武蔵野大学薬学部薬学科有機合成化学研究室

発表論文

2024

"Fentanyl Analogs Exert Antinociceptive Effects via Sodium Channel Blockade in Mice"

Kasai, S.; Ogawa, N.; Takagi, M.; Takahashi, Y.; Makino, K.; Arita, H.; Takahashi, H.; Yoshizawa, K.
Biol. Pharm. Bull. 2024, 47, 872-877. DOI: 10.1248/bpb.b24-00048


"Divergent synthesis of multi-substituted phenanthrenes via an internal redox reaction/ring expansion sequence"

Koyama, R.; Anada, M.; Sueki, S.; Makino, K.; Kojima, T.; Kawasaki-Takasuka, T.; Mori, K.
Chem. Commun. 2024, 60, 3822-3825. DOI: 10.1039/d4cc00797b


"Total Synthesis of Alanense A through an Intramolecular Friedel–Crafts Alkylation"

Makino, K.; Fukuda, R.; Sueki, S.; Anada, M.
J. Org. Chem. 2024, 89, 2050-2054. DOI: 10.1021/acs.joc.3c02481
Selected as Cover Picture.

"Physiologically based pharmacokinetic model analysis of the inhibitory effect of vonoprazan on the metabolic activation of proguanil"

Okubo, K.; Kudo, T.; Yoshihara, S.; Nakabayashi, Y.; Nakauchi, K.; Tanaka, A.; Saito, M.; Tsujisawa, A.; Goda, H.; Yamagishi, Y.; Otake, C.; Makino, K.; Takahashi, H.; Ito, K.
Drug Metab. Pharmacokinet. 2024, 54, 100537. DOI: 10.1016/j.dmpk.2023.100537

2023

"An application of the magnetometer detection system to Crl:CD1 (ICR) mice for head twitch response induced by hallucinogenic 5-HT2A agonists"

Nakamura, M.; Hojo, M.; Kawai, A.; Ikushima, K.; Nagasawa, A.; Takahashi, H.; Makino, K.; Suzuki, T.; Suzuki, J.; Inomata, A.
Fundam. Toxicol. Sci. 2023, 10, 189-197. DOI: 10.2131/fts.10.189

"Drugs possessing aryloxypropanamine pharmacophore, duloxetine, dapoxetine and propranolol, increase allopregnanolone in rat brain: Possible involvement of allopregnanolone in their central nervous system effects"

Nishimoto-Kusunose, S.; Hirakawa, A.; Tanaka, A.; Yoshizawa, K.; Makino, K.; Takahashi, H.; Higashi T.
Steroids 2023, 198, 109272-109280. DOI: 10.1016/j.steroids.2023.109272

"Stereochemistry of N-acyl 5H-dibenzo[b,d]azepne-7(6H)-ones"

Chiba, A.; Tanaka, R.; Hotta, M.; Nakamura, K.; Makino, K.; Tabata, H.; Oshitari, T.; Natsugari, H.; Takahashi, H.
Molecules 2023, 28, 4374-4385. DOI: 10.3390/molecules28124734

"Cytotoxic effects of psychoactive isobutyrylfentanyl and its halogenated derivatives on isolated rat hepatocytes"

Nakagawa, Y.; Suzuki, J.; Suzuki, T.; Takahashi, H.; Makino, K.; Ono, Y.; Sakamoto, M.; Inomata, A.
J. Appl. Toxicol. 2023, in press. DOI: 10.1002/jat.4472

"Stereochemical Analysis of Trifluoroacetamide Derivatives Based on Through-Space 1H−19F Spin−Spin Couplings"

Li, Y.; Ohtake, C.; Hotta, M.; Tabata, H.; Hirano, K.; Iida, M.; Nakamura, K.; Makino, K.; Oshitari, T.; Natsugari, H.; Kusumi, T.; Takahashi H.
J. Org. Chem. 2023, 88, 7026-7037. DOI: 10.1021/acs.joc.3c00311


"Conversion of Racemic Alkyl Aryl Sulfoxides into Pure Enantiomers Using a Recycle Photoreactor: Tandem Use of Chromatography on Chiral Support and Photoracemization on Solid Support"

Tozawa, K.; Makino, K.; Tanaka, Y.; Nakamura, K.; Inagaki, A.; Tabata, H.; Oshitari, T.; Natsugari, H.; Kuroda, N.; Kanemaru, K.; Oda, Y.; Takahashi, H.
J. Org. Chem. 2023, 88, 6955-6961. DOI: 10.1021/acs.joc.3c00265


"Brønsted Acid-Catalyzed Intramolecular 7-endo Hydroarylation Reaction of 1,5-Diaryl-1-pentynes"

Makino, K.; Sueki, S.; Anada, M.
Adv. Synth. Catal. 2023, 365, 1471-1476. DOI: 10.1002/adsc.202300220


"Direct Access to 9/6-Fused Cycles via Sequential Hydride Shift Mediated Double C(sp3)−H Bond Functionalization"

Nakamura, I.; Anada, M.; Sueki, S.; Makino, K.; Mori, K.
Adv. Synth. Catal. 2023, 365, 502-507. DOI: 10.1002/adsc.202201354


"Hepatic and renal toxicities and metabolism of fentanyl analogues in rats"

Ono, Y.; Sakamoto, M.; Makino, K.; Tayama, K.; Tada, Y.; Nakagawa, Y.; Nakajima, J.; Suzuki, J.; Suzuki, T.; Takahashi, H.; Inomata, A.; Moriyasu, T.
Naunyn-Schmiedeb. Arch. Pharmacol. 2023, 396, 149–159. DOI: 10.1007/s00210-022-02301-8


2022

"Inhibition of the chemokine signal regulator FROUNT by disulfiram ameliorates crescentic glomerulonephritis"

Toda, E.; Sawada, A.; Takeuchi, K.; Wakamatsu, K.; Ishikawa, A.; Kuwahara, N.; Sawa, Y.; Hatanaka, S.; Kokubo, K.; Makino, K.; Takahashi, H.; Endo, Y.; Kunugi, S.; Terasaki, M.; Terasaki, Y.; Matsushima, K.; Terashima, Y.; Shimizu, A.
Kidney Int. 2022, 102, 1276–1290. DOI: 10.1016/j.kint.2022.07.031


"Trajectory of the spectral/structural rearrangements for photo-oxidative reaction of neat ketoprofen and its cyclodextrin complex"

Hiroshige, R.; Goto, S.; Tsunoda, C.; Ichii, R.; Shimizu, S.; Otsuka, Y.; Makino, K.; Takahashi, H.; Yokoyama, H.
J. Incl. Phenom. Macrocycl. Chem. 2022, 102, 791–800. DOI: 10.1007/s10847-022-01160-3


"Atropisomeric Properties of N-Alkyl/Aryl 5H-Dibenz[b,f]azepines"

Tanaka, R.; Nabae, A.; Yamane, K.; Makino, K.; Tabata, H.; Oshitari, T.; Natsugari, H.; Takahashi, H.
Chem. Pharm. Bull. 2022, 70, 573-579. DOI: 10.1248/cpb.c22-00265


"Axial chirality and affinity at the GABAA receptor of triazolobenzodiazepines"

Tanaka, R.; Makino, K.; Tabata, H.; Oshitari, T.; Natsugari, H.; Takahashi, H.
Bioorg. Med. Chem. 2022, 64, 116758-116767. DOI: 10.1016/j.bmc.2022.116758


"Photoisomerization of Sulindac and Ozagrel Hydrochloride by Vitamin B2 Catalyst Under Visible Light Irradiation"

Suga, M.; Makino, K.; Tabata, H.; Oshitari, T.; Natsugari, H.; Takahashi, H.
Pharm. Res. 2022, 39, 577-586. DOI: 10.1007/s11095-022-03203-3


"Disulfiram Produces Potent Anxiolytic-Like Effects Without Benzodiazepine Anxiolytics-Related Adverse Effects in Mice"

Saitoh, A.; Nagayama, Y.; Yamada, D.; Makino, K.; Yoshioka, T.; Yamanaka, N.; Nakatani, M.; Takahashi, Y.; Yamazaki, M.; Shigemoto, C.; Ohashi, M.; Okano, K.; Omata, T.; Toda, E.; Sano, Y.; Takahashi, H.; Matsushima, K.; Terashima, Y.
Front. Pharmacol. 2022, 13, 826783. DOI: 10.3389/fphar.2022.8267839


"Protective effects of cyclodextrins on edaravone degradation induced by atmospheric oxygen or additive oxidant"

Hiroshige, R.; Goto, S.; Ichii, R.; Shimizu, S.; Wada-Hirai, A.; Li, Y.-P.; Shimada, Y.; Otsuka, Y.; Makino, K.; Takahashi, H.
J. Incl. Phenom. Macrocycl. Chem. 2022, 102, 327–338. DOI: 10.1007/s10847-021-01122-1



2021

"Rapid Photoracemization of Chiral Alkyl Aryl Sulfoxides"

Makino, K.; Tozawa, K.; Tanaka, Y.; Inagaki, A.; Tabata, H.; Oshitari, T.; Natsugari, H.; Takahashi, H.
J. Org. Chem. 2021, 86, 17249–17256. DOI: 10.1021/acs.joc.1c02320



"Singular value decomposition analysis of the secondary structure features contributing to the circular dichroism spectra of model proteins"

Shiratori, T.; Goto, S.; Sakaguchi, T.; Kasai, T.; Otsuka, Y.; Higashi, K.; Makino, K.; Takahashi, H.; Komatsu, K.
Biochem. Biophys. Rep. 2021, 28, 101153. DOI: 10.1016/j.bbrep.2021.101153


"Experimental Study on the Raman Spectra of Imine Emulsification with Chemometrics"

Otsuka, Y.; Makino, K.; Takahashi, H.
J. Oleo Sci. 2021, 53, 4682-4688. DOI: 10.5650/jos.ess21073


"Atropisomeric Properties of 9-Methyl-1,4-benzodiazepin-2-ones"

Ryoko, T.; Makino, K.; Tabata, H.; Oshitari, T.; Natsugari, H.; Takahashi, H.
Synthesis 2021, 53, 4682-4688. DOI: 10.1055/s-0040-1720865



"Pharmacokinetics of CuGTSM, a Novel Drug Candidate, in a Mouse Model of Menkes Disease"

Yamagishi, Y.; Kudo, T.; Oyumi, M.; Sakamoto, Y.; Takahashi, K.; Akashi, T.; Kobayashi, S.; Kawakami, T.; Goda, H.; Sato, Y.; Mimaki, M.; Kodama, H.; Munakata, M.; Makino, K.; Takahashi, H.; Fukami, T.; Ito, K.
Pharm. Res. 2021, 38, 1335-1344. DOI: 10.1007/s11095-021-03090-0


"Differences in the antinociceptive effects of serotonin–noradrenaline reuptake inhibitors via sodium channel blockade using the veratrine test in mice"

Yoshizawa, K.; Suzuki, Y.; Nakamura, T.; Takahashi, Y.; Makino, K.; Takahashi, H.
Neuroreport 2021, 32, 792-802. DOI: 10.1097/WNR.0000000000001658


"Atropisomeric Properties of N-Acyl/N-Sulfonyl 5H-Dibenzo[b,d]azepin-7(6H)-ones"

Namba, T.; Hotta, M.; Tabata, H.; Makino, K.; Oshitari, T.; Natsugari, H.; Takahashi, H.
J. Org. Chem. 2021, 86, 7563–7578. DOI: 10.1021/acs.joc.1c00594



"Conformational Preference of 2′-Fluoro-Substituted Acetophenone Derivatives Revealed by Through-Space 1H–19F and 13C–19F Spin–Spin Couplings"

Otake, C.; Namba, T.; Tabata, H.; Makino, K.; Hirano, K.; Oshitari, T.; Natsugari, H.; Kusumi, T.; Takahashi, H.
J. Org. Chem. 2021, 86, 4638-4645. DOI: 10.1021/acs.joc.1c00051



"Diastereo- and Enantioselective Intramolecular 1,6-C–H Insertion Reaction of Diaryldiazomethanes Catalyzed by Chiral Dirhodium(II) Carboxylates"

Ito, M.; Kondo, Y.; Namie, R.; Natori, Y.; Takeda, K.; Nambu, H.; Anada, M.; Yamamoto, Y.; Hashimoto, S.
HeteroCycles 2021, 103, 1078-1098. DOI: 10.3987/COM-20-S(K)61



2020

"Chiral paddle-wheel diruthenium complexes for asymmetric catalysis"

Miyazawa, T.; Suzuki, T.; Kumagai, Y.; Takizawa, K.; Kikuchi, T.; Kato, S.; Onoda, A.; Hayashi, T.; Kamei, Y.; Kamiyama, F.; Anada, M.; Kojima, M.; Yoshino, Y.; Matsunaga, S.
Nat. Catal. 2020, 3, 851-858. DOI: 10.1038/s41929-020-00513-w




2019

"Unveiling Two Consecutive Hydroxylations: Mechanisms of Aromatic Hydroxylations Catalyzed by Flavin‐Dependent Monooxygenases for the Biosynthesis of Actinorhodin and Related Antibiotics"

Hashimoto, M.; Taguchi, T.; Ishikawa, K.; Mori, R.; Hotta, A.; Watari, S.; Katakawa, K.; Kumamoto, T.; Okamoto, S.; Ichinose, K.
ChemBioChem 2019, 21, 623. DOI: 10.1002/cbic.201900490
Selected as cover picture


"Isolation of Sesquiterpene–Amino Acid Conjugates, Onopornoids A–D, and a Flavonoid Glucoside from Onopordum alexandrinum"

Sugimoto, S.; Yamano, Y.; Desoukey, S. Y.; Katakawa, K.; Wanas, A. S.; Otsuka, H.; Matsunami, K.
J. Nat. Prod. 2019, 82, 1471. DOI: 10.1021/acs.jnatprod.8b00948


"Direct C4-Benzylation of Indoles via Tandem Benzyl Claisen/Cope Rearrangements"

Abe, T.; Kosaka, Y.; Harasawa, M.; Mishina, A.; Nagasue, M.; Sugimoto, Y.; Katakawa, K.; Sueki, S.; Anada, M.; Yamada, K.
Org. Lett. 2019, 21, 826. DOI: 10.1021/acs.orglett.8b04120


2018

"5-((3-Bromoallyl)Sulfonyl)-1H-Tetrazoles for Bromodiene Synthesis"

Miyazawa, T.; Minami, K.; Ito, M;, Anada, M.; Matsunaga, S.; Hashimoto, S.
HeteroCycles 2018, 97, 1304. DOI: 10.3987/COM-18-S(T)90


"Design, synthesis, and evaluation of polyamine-memantine hybrids as NMDA channel blockers"

Kumamoto, K.; Nakajima, M.; Uga, R.; Iharazaka, N.; Kashihara, H.; Katakawa, K.; Ishikawa, T.; Saiki, R.; Nishimura, K.; Igarashi, K.
Bioorg. Med. Chem. 2018, 26, 603. DOI: 10.1016/j.bmc.2017.12.021


"抗HIV活性三量体ベンゾクロメンConocurvoneとその単量体の化学:単量体Teretifolione Bとその関連化合物の合成研究"

片川 和明, 熊本 卓哉
有機合成化学協会誌 2018, 76, 722. DOI: 10.5059/yukigoseikyokaishi.76.722

"Facile, Efficient Synthesis of Star-Shaped π-Conjugated Systems by Combined Olefin Metathesis with Wittig-type Coupling"

Fujio, T.; Miwata, T.; Takase, M.; Sueki, S.; Nomura, K.
J. Chin. Chem. Soc. 2018, 65, 317. DOI: 10.1002/jccs.201700058

"Preparation of Optically Active 2,2-Disubstituted 5-Hydroxychromenes by the Enzymatic Resolution of Racemic Esters"

Kainuma, M.; Yamada, A.; Katakawa, K.; Kumamoto, T.
HeteroCycles 2018, 97, 604. DOI: 10.3987/COM-18-S(T)45


2017

"Structural and thermodynamic analyses reveal critical features of glycopeptide recognition by the human PILRα immune cell receptor"

Furukawa, A.; Kakita, K.; Yamada, T.; Ishizuka, M.; Sakamoto, J.; Hatori, N.; Maeda, N.; Ohsaka, F.; Saitoh, T.; Nomura, T.; Kuroki, K.; Nambu, H.; Arase, H.; Matsunaga, S.; Anada, M.; Ose, T.; Hashimoto, S.; Maenaka, K.
J. Biol. Chem. 2017, 292, 21128. DOI: 10.1074/jbc.M117.799239

"Total Synthesis of Brasilicardins A and C"

Anada M.; Hanari T.; Kakita K.; Kurosaki Y.; Katsuse K.; Sunadoi Y.; Jinushi Y.; Takeda K.; Matsunaga S.; Hashimoto S.
Org. Lett. 2017, 19, 5581. DOI: 10.1021/acs.orglett.7b02728


"2-Hydroxyindoline-3-triethylammonium Bromide: A Reagent for Formal C3-Electrophilic Reactions of Indoles"

Abe T.; Suzuki, T.; Anada M.; Matsunaga, S.; Yamada K.
Org. Lett. 2017, 19, 4275. DOI: 10.1021/acs.orglett.7b01940


"Catalytic Enantioselective Desymmetrization of meso-Aziridines with Fluoromalonates"

Fukagawa, S.; Xu, Y.; Anada, M.; Yoshino, T.; Matsunaga, S.
HeteroCycles 2017, 94, 1337. DOI: 10.3987/COM-17-13725


"Diastereo- and Enantioselective Construction of 6,7-Dioxabicyclo[2.2.1]heptane Derivatives by a Dirhodium(II)-Catalyzed Intramolecular C-H Insertion Reaction"

Miyazawa, T.; Imai, K.; Ito, M.; Takeda, K.; Anada, M.; Matsunaga, S.; Hashimoto, S.
HeteroCycles 2017, 95, 1211. DOI: 10.3987/COM-16-S(S)72


"Asymmetric total syntheses of teretifolione B and methylteretifolione B via Diels-Alder reaction of optically active pyranobenzyne and substituted furans"

Katakawa, K.; Kainuma, M.; Suzuki, K.; Tanaka, S.; Kumamoto, T.
Tetrahedron 2017, 73, 5063. DOI: 10.1016/j.tet.2017.06.050


"Total synthesis of (+)-blennolide C and (+)-gonytolide C via spirochromanone"

Adachi, K.; Hasegawa, S.; Katakawa, K.; Kumamoto, T.
Tetrahedron Lett. 2017, 58, 4479. DOI: 10.1016/j.tetlet.2017.10.038


"Synthesis of Poly(arylene vinylene)s Containing Different End Groups by Combined Acyclic Diene Metathesis Polymerization with Wittig-type Couplings"

Miyashita, T.; Kunisawa, M.; Sueki, S.; Nomura, K.
Angew. Chem. Int. Ed. 2017, 56, 5288. DOI: 10.1002/anie.201700466
Selected as inside back cover


"Effect of Al Cocatalyst in Ethylene Polymerization by (Imido)vanadium Dichloride Complexes Containing Anionic N-Heterocyclic Carbenes Having a Weakly Coordinating Borate Moiety"

Nagai, G.; Mitsudome, T.; Tsutsumi, K.; Sueki, S.; Ina, T.; Tamm. M.; Nomura, K.
J. Jpn. Petrol. Inst. 2017, 60, 256. DOI: 10.1627/jpi.60.256


2016

"Rapid Screening by Cell-Based Fusion Assay for Identifying Novel Antivirals of Glycoprotein B-Mediated Herpes Simplex Virus Type 1 Infection"

Maeda, N.; Furukawa, A; Kakita, K.; Anada, M.; Hashimoto, S.; Matsunaga, S.; Kuroki, K.; Ose, T.; Kato, A.; Arii, J.; Kawaguchi, Y.; Arase, H.; Maenaka, K.
Biol. Pharm. Bull. 2016, 39, 1897. DOI: 10.1248/bpb.b16-00533
Selected as the Cover Picture

"Enantio-and diastereoselective desymmetrization of α-alkyl-α-diazoesters by dirhodium(II)-catalyzed intramolecular C-H insertion"

Miyazawa, T.; Minami, K.; Ito, M;, Anada, M.; Matsunaga, S.; Hashimoto, S.
Tetrahedron 2016, 72, 3939. DOI: 10.1016/j.tet.2016.05.015



"Rhenium-Catalyzed Synthesis of 1,3-Diiminoisoindolines via Insertion of Carbodiimides into a C−H Bond of Aromatic and Heteroaromatic Imidates"

Wang, Z.; Sueki, S.; Kanai, M.; Kuninobu, Y.
Org. Lett. 2016, 18, 2459. DOI: 10.1021/acs.orglett.6b01012


2015

"Asymmetric Total Synthesis of (–)-Englerin A through Catalytic Diastereo- and Enantioselective Carbonyl Ylide Cycloaddition"

Hanari, T.; Shimada, N.; Kurosaki, Y.; Thrimurtulu, N.; Nambu, H.; Anada, M.; Hashimoto, S.
Chem. Eur. J. 2015, 21, 11671. DOI: 10.1002/chem.201502009


"Catalytic Asymmetric Synthesis of (–)-E-δ-Viniferin via an Intramolecular C–H Insertion of Diaryldiazomethane Using Rh2(S-TFPTTL)4"

Natori, Y.; Ito, M.; Anada, M.; Nambu, H.; Hashimoto, S.
Tetrahedron Lett. 2015, 56, 4324. DOI: 10.1016/j.tetlet.2015.05.072


"Diastereo- and Enantioselective Intramolecular 1,6-C–H Insertion Reactions of α-Diazo Esters Catalyzed by Chiral Dirhodium(II) Carboxylates"

Ito, M.; Kondo, Y.; Nambu, H.; Anada, M.; Takeda, K.; Hashimoto, S.
Tetrahedron Lett. 2015, 56, 1397. DOI: 10.1016/j.tetlet.2015.01.125


"An Insight into Different Stabilization Mechanisms of Phenytoin Derivatives Supersaturation by HPMC and PVP"

Otsuka, N.; Ueda, K.; Ohyagi, N.; Shimizu, K.; Katakawa, K.; Kumamoto, T.; Higashi, K.; Yamamoto, K.; Moribe, K.
J. Pharm. Sci. 2015, 104, 2574. DOI: 10.1002/jps.24527

"Rhodium-catalysed synthesis of multi-substituted silylindenes from aryl alkynes and hydrosilanes via C-H bond activation"

Sueki, S.; Kuninobu, Y.
Chem. Commun. 2015, 51, 7685. DOI: 10.1039/c5cc01569c


2014

"Enantio- and Diastereoselective Hetero-Diels–Alder Reactions between 4-Methyl-substituted Rawal’s Diene and Aldehydes Catalyzed by Chiral Dirhodium(II) Carboxamidates: Catalytic Asymmetric Synthesis of (–)-cis-Aerangis Lactone."

Watanabe, Y.; Shimada, N.; Anada, M.; Hashimoto, S.
Tetrahedron: Asymmetry 2014, 25, 63. DOI: 10.1016/j.tetasy.2013.10.016


"Synthesis of a Natural Chromenoquinone via the Diels-Alder Reaction of Pyranobenzyne and Furan"

Katakawa, K.; Sato, A.; Iwasaki, M.; Horikawa, T.; Kumamoto, T.
Chem. Pharm. Bull. 2014, 62, 820. DOI: 10.1248/cpb.c14-00228

"Selective Synthesis of Benzyl Enol Ethers of β-Dicarbonyl Compounds in Basic Condition and the Application Towards Synthesis of Naphthoquinones"

Katakawa, K.; Yonenaga, D.; Terada, N.; Sakamoto, A.; Hoshino, K.; Kumamoto, T.
HeteroCycles 2014, 88, 817. DOI: 10.3987/COM-13-S(S)66


"Synthesis of 1,4-Dihydropyridines and Their Fluorescence Properties"

Sueki, S.; Takei, R.; Zaitsu, Y.; Abe, J.; Fukuda, A.; Seto, K.; Furukawa, Y.; Shimizu, I.
Eur. J. Org. Chem. 2014, 5281. DOI: 10.1002/ejoc.201402426


2013

"Enantioselective Cycloaddition of Carbonyl Ylides with Arylallenes using Rh2(S-TCPTTL)4."

Krishnamurthi, J.; Nambu, H.; Takeda, K.; Anada, M.; Yamano, A.; Hashimoto, S.
Org. Biomol. Chem. 2013, 11, 5374. DOI: 10.1039/C3OB41236A


"Rhenium-Catalyzed Synthesis of 3-Imino-1-isoindolinones via C-H Bond Activation and Its Application to Synthesis of Polyimide Derivatives"

Shunsuke, S.; Guo, Y.; Kanai, M.; Kuninobu, Y.
Angew. Chem. Int. Ed. 2013, 52, 11879. DOI: 10.1002/anie.201306360

Highlights: Synfacts 2014, 10, 34. DOI: 10.1055/s-0033-1340389

"Copper-Catalyzed N- and O-Alkylation of Amines and Phenols using Alkylborane Reagents"

Shunsuke, S.; Kuninobu, Y.
Org. Lett. 2013, 15, 1544. DOI: 10.1021/ol400323z


2012

"Enantio- and Diastereoselective Hetero-Diels-Alder Reactions between 2-Aza-3-silyloxy-1,3-butadienes and Aldehydes Catalyzed by Chiral Dirhodium(II) Carboxamidates"

Watanabe, Y.; Washio, T.; Krishnamurthi, J.; Anada, M.; Hashimoto, S.
Chem. Commun. 2012, 48, 6969. DOI: 10.1039/C2CC32876C


"A Polymer-Supported Chiral Fluorinated Dirhodium(II) Complex for Asymmetric Amination of Silyl Enol Ethers"

Oohara, T.; Nambu, H.; Anada, M.; Takeda, K.; Hashimoto, S.
Adv. Synth. Catal. 2012, 354, 2331. DOI: 10.1002/adsc.201200219


"Catalytic Asymmetric Intermolecular C-H Insertion Reactions of 1,4-Cyclohexadiene with 2,4-Dimethyl-3-pentyl α-Alkyl-α-diazoacetates using Chiral Dirhodium(II) Carboxylates"

Goto, T.; Onozuka, T.; Kosaka, Y.; Anada, M.; Takeda, K.; Hashimoto, S.
HeteroCycles 2012, 86, 1647. DOI: 10.3987/COM-12-S(N)120


2011

"Highly Enantioselective Cyclopropenation Reaction of 1-Alkynes with α-Alkyl-α-diazoesters Catalyzed by Dirhodium(II) Carboxylates"

Goto, T.; Takeda, K.; Shimada, N.; Nambu, H.; Anada, M.; Shiro, M.; Ando, K.; Hashimoto, S.
Angew. Chem, Int. Ed. 2011, 50, 6803. DOI: 10.1002/anie.201101905


"Enantio- and Diastereoselective Cyclopropanation with tert-Butyl α-Diazopropionate Catalyzed by Dirhodium(II) Tetrakis[N-tetrabromophthaloyl-(S)-tert-leucinate]"

Goto, T.; Takeda, K.; Anada, M.; Ando, K.; Hashimoto, S.
Tetrahedron Lett. 2011, 52, 4200. DOI: 10.1016/j.tetlet.2011.06.008


"Ten new fawcettimine-related alkaloids from three species of Lycopodium"

Katakawa, K.; Mito, H.; Kogure, N.; Kitajima, M.; Wongseripipatana, S.; Arisawa, M.; Takayama, H.
Tetrahedron 2011, 67, 6561. DOI: 10.1016/j.tet.2011.05.107



総説・著書・解説・特許


2022

2021

"第8章 質量分析法"

穴田 仁洋
コアカリ対応 分析化学 第4版, 今井 一洋, 荒川 秀俊, 小林 典裕 編, 2021, 丸善出版, 313. (Book Chapter)

"10章 免疫・アレルギー疾患とその治療薬および抗炎症薬"

穴田 仁洋
現場で役に立つ!臨床医薬品化学, 臨床医薬品化学研究会 編, 2021, 化学同人, 186. (Book Chapter)

2020

"キラル多核金属錯体を用いる触媒的不斉合成"

松永 茂樹,穴田 仁洋
CSJ カレントレビュー37「高機能性金属錯体が拓く触媒科学 革新的分子変換反応の創出をめざして」, 日本化学会 編, 2020, 化学同人, 108. (Book Chapter)

"Chemistry of anti-HIV active trimeric pyranonaphtho-quinone conocurvone: Synthetic studies towards monomeric teretifolione B and related compounds"

Kumamoto, K.; Katakawa, K.
Heterocycles, 2020, 100, 177. DOI: 10.3987/REV-19-915


"Manganese Catalysis"

Kuninobu, Y.; Sueki, S.; Ackermann, L.; Kaplaneris, K.
Catalysis with Earth-Abundant Elements, Schneider, U.; Thomas, S. (Eds.), 2020, Royal Society of Chemistry, 139. (Book Chapter) DOI: 10.1039/9781788012775-00139


2019

"ロジウム(II)錯体をルイス酸触媒として用いる不斉ヘテロDiels–Alder反応"

穴田 仁洋, 橋本 俊一
有機合成化学協会誌, 2019, 77, 553. DOI: 10.5059/yukigoseikyokaishi.77.553

"Recent Progress in Aryne Cycloaddition Reactions"

Kumamoto, K.; Katakawa, K.
Cycloaddition Reaction, D. Margetic (Eds.), 2019, Nova Science Publishers, 1. (Book Chapter)

2018

2017

"第5章 アルカロイドの分類と生合成の概要"

片川 和明
アルカロイドの科学 生物活性を生みだす物質の探索から創薬の実際まで, 高山 廣光 編, 2017, 化学同人, 103. (Book Chapter)

"オーファン受容体のリガンド探索が副作用軽減の鍵!?"

片川 和明
ファルマシア 2017, 53, 1211. DOI: 10.14894/faruawpsj.53.12_1211

"酸化剤の一工夫で形勢逆転: Pd触媒によるベンズアゼチジン合成法"

末木 俊輔
ファルマシア 2017, 53, 358. DOI: 10.14894/faruawpsj.53.4_358.

2016

"Recent Progress in Synthesis of Dihydropyridines"

Sueki, S.; Shimizu, I.
New Research on Dihydropyridines, J. Morales (Eds.), 2016, Nova Science Publishers, 1. (Book Chapter)

2015

"C-H Bond Transformations Leading to the Synthesis of Organic Functional Materials"

Kuninobu, Y.; Sueki, S.
Synthesis 2015, 47, 3823. DOI: 10.1055/s-0035-1560346
Selected as the Cover Picture

"Imino-Containing Solvent-Soluble Polyimides, Their Manufacture, and Diimidates Therefor"

Kuninobu, Y.; Sueki, S.
PCT Int. Appl. 2015, JP 2015025061 A 20150205.

2014

"Propanoic acid, 2-Diazo-, 2-methyl-1-(1-methylethyl)propyl ester"

Anada, M.; Takeda, K.; Ito, M.; Hashimoto, S.
e-EROS Encyclopedia of Reagents for Organic Synthesis, 2014. DOI: 10.1002/047084289X.rn01693


2013

2012

"分子状酸素を用いる炭素-酸素結合生成反応—効率的な酸素官能基導入反応—"

末木 俊輔
有機合成化学協会誌, 2012, 70, 71. DOI: 10.5059/yukigoseikyokaishi.70.71

2011

"触媒的C-H活性化を機軸とする天然物合成"

穴田 仁洋,南部 寿則,橋本 俊一
CSJ カレントレビュー05「不活性結合・不活性分子の活性化 革新的な分子変換反応の開拓」, 日本化学会編, 2011, 化学同人, 175. (Book Chapter)

"天然有機化合物の分離・精製, 化学構造解析"

大川 雅史, 大塚 功, 片川 和明, 川口 基一郎, 北中 進, 高松 智, 平井 康明, 平野 裕之, 船山 信次, 安田 高明
医療を指向する天然物医薬品化学 第2版, 北中 進, 船山 信次 編, 2011, 廣川書店, 115. (Book Chapter)

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